SCHEMBL19937622

SCHEMBL19937622

COc1cc(-c2ccn(C3CCC3)n2)cnc1N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 7/20 0.52
INSR P06213 1/20 0.50
NPM1 P06748 1/20 0.50
ALK Q9UM73 1/20 0.50
MAP3K11 Q16584 1/20 0.49
PIK3CA P42336 6/20 0.43
PIK3CD O00329 5/20 0.43
PIK3CG P48736 5/20 0.43
ABL1 P00519 3/20 0.43
EGFR P00533 3/20 0.43
HCK P08631 3/20 0.43
SRC P12931 3/20 0.43
KDR P35968 3/20 0.43
PIK3CB P42338 3/20 0.43
MTOR P42345 3/20 0.43
EPHB4 P54760 3/20 0.43
PRKDC P78527 3/20 0.43
PI4KB Q9UBF8 3/20 0.43
FGFR1 P11362 2/20 0.42
FGFR2 P21802 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19937634 0.98 MAP3K11 (0.52) MAP3K12INSRNPM1ALKMAP3K11
SCHEMBL19937772 0.87 INSR (0.57) MAP3K12INSRNPM1ALKJAK2
SCHEMBL19937630 0.85 INSR (0.57) MAP3K12INSRNPM1ALKJAK2
SCHEMBL19937609 0.85 INSR (0.54) MAP3K12INSRNPM1ALK
SCHEMBL19937624 0.85 MAP3K12 (0.54) MAP3K12INSRNPM1ALK
SCHEMBL19937632 0.82 MAP3K12 (0.54) MAP3K12INSRNPM1ALK
SCHEMBL19937777 0.82 INSR (0.54) MAP3K12INSRNPM1ALK
SCHEMBL19937610 0.81 MAP3K12 (0.51) MAP3K12INSRNPM1ALK
SCHEMBL19937643 0.80 MAP3K12 (0.50) MAP3K12INSRNPM1ALKFGFR1
SCHEMBL19937789 0.79 INSR (0.42) MAP3K12INSRNPM1ALKMAP3K11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2945938-B1 3-SUBSTITUTED PYRAZOLES AND USE AS DLK INHIBITORS HOFFMANN LA ROCHE (CH) 2018-03-07 EP disclosed