SCHEMBL19937772

SCHEMBL19937772

CC(C)Oc1cc(-c2ccn(C3CCC3)n2)cnc1N

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
INSR P06213 1/20 0.57
NPM1 P06748 1/20 0.57
ALK Q9UM73 1/20 0.57
MAP3K12 Q12852 13/20 0.54
JAK2 O60674 3/20 0.47
MET P08581 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19937630 0.98 INSR (0.57) INSRNPM1ALKMAP3K12JAK2
SCHEMBL19937609 0.89 INSR (0.54) INSRNPM1ALKMAP3K12
SCHEMBL19937622 0.87 MAP3K12 (0.52) INSRNPM1ALKMAP3K12JAK2
SCHEMBL19937777 0.86 INSR (0.54) INSRNPM1ALKMAP3K12
SCHEMBL19937634 0.85 MAP3K11 (0.52) INSRNPM1ALKMAP3K12JAK2
SCHEMBL19937624 0.82 MAP3K12 (0.54) INSRNPM1ALKMAP3K12
SCHEMBL19937632 0.80 MAP3K12 (0.54) INSRNPM1ALKMAP3K12
SCHEMBL19937610 0.78 MAP3K12 (0.51) INSRNPM1ALKMAP3K12
SCHEMBL19937588 0.78 MAP3K12 (0.47) INSRNPM1ALKMAP3K12JAK2
SCHEMBL19937762 0.78 MAP3K12 (0.52) INSRNPM1ALKMAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2945938-B1 3-SUBSTITUTED PYRAZOLES AND USE AS DLK INHIBITORS HOFFMANN LA ROCHE (CH) 2018-03-07 EP disclosed