SCHEMBL19937632

SCHEMBL19937632

Nc1ncc(-c2ccn(C3CCCC3)n2)cc1OC(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 19/20 0.54
INSR P06213 1/20 0.48
NPM1 P06748 1/20 0.48
ALK Q9UM73 1/20 0.48
MAP3K13 O43283 1/20 0.45
STK16 O75716 1/20 0.45
PAK4 O96013 1/20 0.45
NTRK1 P04629 1/20 0.45
FLT3 P36888 1/20 0.45
MAP3K9 P80192 1/20 0.45
MAP3K10 Q02779 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19937624 0.98 MAP3K12 (0.54) MAP3K12INSRNPM1ALKMAP3K13
SCHEMBL19937634 0.85 MAP3K11 (0.52) MAP3K12INSRNPM1ALK
SCHEMBL19937777 0.84 INSR (0.54) MAP3K12INSRNPM1ALK
SCHEMBL19937622 0.82 MAP3K12 (0.52) MAP3K12INSRNPM1ALK
SCHEMBL19937751 0.82 MAP3K12 (0.53) MAP3K12
SCHEMBL19937609 0.82 INSR (0.54) MAP3K12INSRNPM1ALK
SCHEMBL19937630 0.82 INSR (0.57) MAP3K12INSRNPM1ALK
SCHEMBL19937642 0.80 MAP3K12 (0.55) MAP3K12
SCHEMBL19937762 0.80 MAP3K12 (0.52) MAP3K12INSRNPM1ALK
SCHEMBL19937772 0.80 INSR (0.57) MAP3K12INSRNPM1ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2945938-B1 3-SUBSTITUTED PYRAZOLES AND USE AS DLK INHIBITORS HOFFMANN LA ROCHE (CH) 2018-03-07 EP disclosed