SCHEMBL19944409

SCHEMBL19944409

Cc1ccc(F)c(C(N)=O)c1OCCCCN1CC=C(c2ccc(F)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.49
SIGMAR1 Q99720 7/20 0.47
CYP2D6 P10635 1/20 0.46
THPO P40225 1/20 0.46
LMNA P02545 1/20 0.45
PMP22 Q01453 1/20 0.45
PPARG P37231 1/20 0.44
PPARA Q07869 1/20 0.44
PARP1 P09874 1/20 0.42
HTR1A P08908 2/20 0.42
HTR7 P34969 1/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19944866 0.84 PARP1 (0.47) DRD2SIGMAR1CYP2D6THPOLMNA
SCHEMBL19944378 0.75 SIGMAR1 (0.49) DRD2SIGMAR1CYP2D6THPOLMNA
SCHEMBL19944416 0.74 DRD2 (0.61) DRD2SIGMAR1CYP2D6THPOLMNA
SCHEMBL8010714 0.74 SIGMAR1 (0.72) DRD2SIGMAR1PARP1HTR7
SCHEMBL11830521 0.73 SIGMAR1 (0.64) DRD2SIGMAR1PARP1HTR7
SCHEMBL19944499 0.71 SIGMAR1 (0.47) DRD2SIGMAR1PPARGPPARAPARP1
SCHEMBL19944762 0.71 SIGMAR1 (0.64) DRD2SIGMAR1PARP1HTR1AHTR7
SCHEMBL8575395 0.69 SIGMAR1 (0.62) DRD2SIGMAR1PARP1HTR7ATM
SCHEMBL28057913 0.69 SIGMAR1 (0.56) DRD2SIGMAR1PPARGPPARAPARP1
SCHEMBL6367176 0.69 DRD2 (0.61) DRD2SIGMAR1CYP2D6THPOLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018044136-A1 NOVEL COMPOUND, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT FOR PREVENTING OR TREATING DISEASES ASSOCIATED WITH POLY(ADP-RIBOSE) POLYMERASE-1 (PARP-1) 충남대학교 산학협력단 2018-03-08 WO disclosed