SCHEMBL19944378

SCHEMBL19944378

NC(=O)c1cccc(N)c1OCCCN1CC=C(c2ccc(F)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.49
DRD2 P14416 3/20 0.48
CYP2D6 P10635 1/20 0.47
THPO P40225 1/20 0.47
HTR6 P50406 2/20 0.47
LMNA P02545 1/20 0.46
PMP22 Q01453 1/20 0.46
HTR7 P34969 1/20 0.45
PARP1 P09874 3/20 0.44
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43
KCNH2 Q12809 1/20 0.43
PARP2 Q9UGN5 1/20 0.43
HTR1A P08908 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19944499 0.90 SIGMAR1 (0.47) SIGMAR1DRD2HTR7PARP1PPARG
SCHEMBL19944416 0.86 DRD2 (0.61) SIGMAR1DRD2CYP2D6THPOHTR6
SCHEMBL19944866 0.86 PARP1 (0.47) SIGMAR1DRD2CYP2D6THPOHTR6
SCHEMBL7295751 0.75 HTR1A (0.57) SIGMAR1DRD2HTR1A
SCHEMBL19944409 0.75 DRD2 (0.49) SIGMAR1DRD2CYP2D6THPOLMNA
SCHEMBL8010714 0.73 SIGMAR1 (0.72) SIGMAR1DRD2HTR7PARP1
SCHEMBL28057913 0.73 SIGMAR1 (0.56) SIGMAR1DRD2HTR7PARP1PPARG
SCHEMBL8909829 0.72 CYP2D6 (0.48) SIGMAR1CYP2D6THPOLMNAPMP22
SCHEMBL7861690 0.71 CYP2D6 (0.71) SIGMAR1CYP2D6THPOLMNAPMP22
SCHEMBL6367176 0.70 DRD2 (0.61) SIGMAR1DRD2CYP2D6THPOLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018044136-A1 NOVEL COMPOUND, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT FOR PREVENTING OR TREATING DISEASES ASSOCIATED WITH POLY(ADP-RIBOSE) POLYMERASE-1 (PARP-1) 충남대학교 산학협력단 2018-03-08 WO disclosed