SCHEMBL19953522

SCHEMBL19953522

CN1C(=O)Cc2ccccc2[C@H]1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACE P12821 6/20 0.47
HDAC4 P56524 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
NOTUM Q6P988 1/20 0.41
SRD5A1 P18405 2/20 0.40
GRM7 Q14831 1/20 0.39
ANPEP P15144 2/20 0.39
PDE5A O76074 1/20 0.38
RNASEH1 O60930 1/20 0.37
HPGD P15428 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
NCOR2 Q9Y618 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953652 1.00 ACE (0.47) ACEHDAC4HDAC7HDAC5NOTUM
SCHEMBL19960636 0.83 HDAC4 (0.43) HDAC4HDAC7HDAC5NOTUMSRD5A1
SCHEMBL19960827 0.81 ANPEP (0.40) ACEHDAC4HDAC7HDAC5NOTUM
SCHEMBL19953701 0.80 ACE (0.47) ACEHDAC4HDAC7HDAC5NOTUM
SCHEMBL19960826 0.80 ACE (0.47) ACEHDAC4HDAC7HDAC5NOTUM
SCHEMBL19953646 0.80 ACE (0.47) ACEHDAC4HDAC7HDAC5NOTUM
SCHEMBL19953669 0.80 MEN1 (0.42) NOTUMHPGD
SCHEMBL19953636 0.79 FABP5 (0.44) HDAC4HDAC7HDAC5GRM7
SCHEMBL19953670 0.78 ACE (0.42) ACEGRM7
SCHEMBL14987797 0.76 SRD5A1 (0.44) HDAC4HDAC7HDAC5NOTUMSRD5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed