SCHEMBL19953529

SCHEMBL19953529

O=C(O)[C@@H]1c2ccccc2CCN1C(=O)C1CC1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACE P12821 6/20 0.61
F11 P03951 1/20 0.56
TSHR P16473 1/20 0.50
ALDH1A1 P00352 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
KEAP1 Q14145 7/20 0.47
MTNR1B P49286 1/20 0.44
NFE2L2 Q16236 3/20 0.44
ATM Q13315 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953642 1.00 ACE (0.61) ACEF11TSHRALDH1A1NPSR1
SCHEMBL19960681 0.87 F11 (0.55) ACEF11TSHRALDH1A1NPSR1
SCHEMBL16111164 0.84 ACE (0.68) ACETSHRNPSR1KEAP1MTNR1B
SCHEMBL19960667 0.83 F11 (0.53) ACEF11TSHRALDH1A1NPSR1
SCHEMBL19953516 0.83 F11 (0.53) ACEF11TSHRALDH1A1NPSR1
SCHEMBL19953782 0.80 F11 (0.55) ACEF11TSHRALDH1A1NPSR1
SCHEMBL19953658 0.80 F11 (0.50) ACEF11TSHRALDH1A1NPSR1
SCHEMBL19953491 0.80 F11 (0.50) ACEF11TSHRALDH1A1NPSR1
SCHEMBL19953756 0.79 F11 (0.48) ACEF11TSHRALDH1A1NPSR1
SCHEMBL10901972 0.78 ACE (0.60) ACEKEAP1MTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed