SCHEMBL19953619

SCHEMBL19953619

CN1C(=O)CC(C(=O)O)c2c(F)cc(F)cc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.34
ALDH1A1 P00352 2/20 0.33
BRD4 O60885 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GAA P10253 2/20 0.33
EPHX2 P34913 1/20 0.33
TSHR P16473 1/20 0.33
POLB P06746 1/20 0.33
PYGL P06737 1/20 0.32
PYGM P11217 1/20 0.32
ESR2 Q92731 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
LMNA P02545 1/20 0.31
HTR1F P30939 1/20 0.31
MAPK1 P28482 1/20 0.31
HSD17B10 Q99714 1/20 0.31
HTR7 P34969 1/20 0.30
HTT P42858 1/20 0.30
DPP4 P27487 1/20 0.30
CYP11B1 P15538 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953762 0.67 ALDH1A1 (0.46) ALDH1A1BRD4SMN1; SMN2GAATSHR
SCHEMBL17919028 0.67 BRD4 (0.34) BRD4
SCHEMBL19953671 0.66 ALDH1A1 (0.39) ALDH1A1BRD4GAATSHRMAPK1
SCHEMBL31277845 0.62 LTB4R (0.33) GAAPOLBHTT
SCHEMBL17144273 0.60 EPHX2 (0.40) EPHX2
SCHEMBL20177699 0.60 FPR2 (0.42)
SCHEMBL10288452 0.60 FFAR1 (0.40) HTT
SCHEMBL10288624 0.60 FFAR1 (0.40) HTT
SCHEMBL2137635 0.60 FFAR1 (0.40) HTT
SCHEMBL19960629 0.59 MEN1 (0.32) ALDH1A1POLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed