SCHEMBL19953667

SCHEMBL19953667

O=C(NC1Cc2ccccc2C1)C1c2ccccc2CCN1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.47
MTNR1B P49286 4/20 0.46
MTNR1A P48039 3/20 0.46
FABP5 Q01469 1/20 0.44
F11 P03951 1/20 0.43
HHAT Q5VTY9 2/20 0.41
GRM7 Q14831 2/20 0.41
HDAC8 Q9BY41 1/20 0.41
CYP2D6 P10635 1/20 0.41
HRH3 Q9Y5N1 2/20 0.40
CASP3 P42574 1/20 0.40
CASP2 P42575 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19960671 0.86 HRH3 (0.47) ACEMTNR1BMTNR1AF11HRH3
SCHEMBL19953782 0.86 F11 (0.55) ACEMTNR1BMTNR1AFABP5F11
SCHEMBL19960670 0.83 GHSR (0.49) MTNR1BMTNR1AFABP5
SCHEMBL19953699 0.82 ACE (0.46) ACEMTNR1BMTNR1AFABP5F11
SCHEMBL16111164 0.80 ACE (0.68) ACEMTNR1BHHAT
SCHEMBL19953578 0.79 ACE (0.41) ACEMTNR1BF11HHATCYP2D6
SCHEMBL19953576 0.79 ACE (0.41) ACEMTNR1BF11HHATCYP2D6
SCHEMBL19953575 0.79 ACE (0.41) ACEMTNR1BF11HHATCYP2D6
SCHEMBL19960664 0.78 HDAC8 (0.43) ACEMTNR1BMTNR1AF11HDAC8
SCHEMBL19960847 0.78 EPHX2 (0.43) ACEMTNR1BMTNR1AFABP5CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed