SCHEMBL19953576

SCHEMBL19953576

CO[C@@H]1c2ccccc2C[C@H]1NC(=O)C1c2ccccc2CCN1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACE P12821 4/20 0.41
CASP3 P42574 1/20 0.39
CASP2 P42575 1/20 0.39
F11 P03951 2/20 0.38
XIAP P98170 4/20 0.38
MTNR1B P49286 1/20 0.38
HHAT Q5VTY9 2/20 0.36
CYP2D6 P10635 1/20 0.36
KLKB1 P03952 1/20 0.35
MMP1 P03956 1/20 0.35
TRPV1 Q8NER1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953575 1.00 ACE (0.41) ACECASP3CASP2F11XIAP
SCHEMBL19953578 1.00 ACE (0.41) ACECASP3CASP2F11XIAP
SCHEMBL19960686 0.89 F11 (0.48) ACECASP3CASP2F11XIAP
SCHEMBL19960811 0.88 GHSR (0.45) XIAP
SCHEMBL19960718 0.86 ACE (0.46) ACECASP3CASP2F11XIAP
SCHEMBL19960692 0.83 ACE (0.44) ACECASP3CASP2F11MTNR1B
SCHEMBL19953667 0.79 ACE (0.47) ACECASP3CASP2F11MTNR1B
SCHEMBL19960812 0.74 TSHR (0.50)
SCHEMBL15355314 0.73 MTNR1B (0.49) ACEMTNR1BHHATCYP2D6TRPV1
SCHEMBL16111164 0.73 ACE (0.68) ACEMTNR1BHHAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed