SCHEMBL19954030

SCHEMBL19954030

OC1(c2ccc3c(c2)CN(I)C3)CCNCC1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.47
DPP4 P27487 1/20 0.41
DPP9 Q86TI2 1/20 0.37
DPP7 Q9UHL4 1/20 0.37
SIGMAR1 Q99720 1/20 0.36
TNF P01375 2/20 0.32
NAMPT P43490 2/20 0.31
MAPKAPK2 P49137 1/20 0.31
OPRM1 P35372 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12853767 0.84 DRD2 (0.47) DRD2DPP4DPP9DPP7SIGMAR1
SCHEMBL19954041 0.81 OPRD1 (0.36) OPRM1
SCHEMBL15247408 0.77 DRD2 (0.53) DRD2SIGMAR1OPRM1
SCHEMBL15247409 0.76 DRD2 (0.40) DRD2DPP4DPP9DPP7SIGMAR1
SCHEMBL30047438 0.75 CRBN (0.57) OPRM1
SCHEMBL5463091 0.70 KCNH2 (0.47) DRD2SIGMAR1
SCHEMBL12853726 0.69 OPRD1 (0.38) OPRM1
SCHEMBL4472985 0.69 DRD2 (0.66) DRD2SIGMAR1MAPKAPK2OPRM1
SCHEMBL2271090 0.68 DRD2 (0.55) DRD2SIGMAR1OPRM1
SCHEMBL654759 0.68 DRD2 (0.65) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9914719-B2 Hydroxybenzamide derivatives and their use as inhibitors of HSP90 ASTEX THERAPEUTICS LTD. (GB) 2018-03-13 US disclosed