SCHEMBL19957732

SCHEMBL19957732

CNc1cnc(N)c(ON)c1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.33
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
SHMT2 P34897 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
FYN P06241 1/20 0.30
AURKA O14965 1/20 0.30
KDR P35968 1/20 0.30
AURKB Q96GD4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7311469 0.74 NOS3 (0.56) DHFRNOS3NOS1NOS2KDM4E
SCHEMBL21712533 0.72 NOS3 (0.34) NOS3NOS1NOS2KDM4EALDH1A1
SCHEMBL21139550 0.69 NOS3 (0.32) NOS3NOS1NOS2KDM4EALDH1A1
SCHEMBL21646346 0.68 IRAK4 (0.33) NOS3NOS1NOS2KDM4EALDH1A1
SCHEMBL20458856 0.68 PIK3CA (0.39) AURKAKDRAURKB
Hydrochloric Acid SCHEMBL30518652 0.67 PIK3CA (0.38) AURKAKDRAURKB
SCHEMBL26739699 0.67 TGFBR1 (0.37) DHFRALDH1A1AURKAAURKB
SCHEMBL24140061 0.65 MAPT (0.50) DHFRKDM4EALDH1A1AURKAKDR
SCHEMBL3936252 0.65 PGK1 (0.43) KDM4EALDH1A1AURKA
SCHEMBL13715975 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2935243-B1 PRMT5 INHIBITORS CONTAINING A DIHYDRO- OR TETRAHYDROISOQUINOLINE AND USES THEREOF EPIZYME INC (US) 2018-03-14 EP disclosed