SCHEMBL19960716

SCHEMBL19960716

CNC(=O)C1c2ccccc2CCN1CC(F)F

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.46
OPRM1 P35372 1/20 0.43
HDAC8 Q9BY41 2/20 0.42
XIAP P98170 6/20 0.41
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
NCOR2 Q9Y618 1/20 0.40
PRMT5 O14744 1/20 0.40
WDR77 Q9BQA1 1/20 0.40
CYP2D6 P10635 2/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
MTNR1B P49286 1/20 0.39
CARM1 Q86X55 1/20 0.39
PRCP P42785 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19960713 0.83 ACE (0.43) ACEOPRM1HDAC8HDAC3HDAC1
SCHEMBL19953503 0.81 OPRM1 (0.43) ACEOPRM1HDAC8HDAC1HDAC2
SCHEMBL19960630 0.81 OPRM1 (0.43) ACEOPRM1HDAC8HDAC1HDAC2
SCHEMBL9744383 0.78 HDAC8 (0.43) ACEOPRM1HDAC8HDAC3HDAC1
SCHEMBL19960810 0.75 PRMT5 (0.43) ACEOPRM1HDAC8HDAC3HDAC1
SCHEMBL19960631 0.70 OPRM1 (0.38) ACEOPRM1XIAPMTNR1B
SCHEMBL4239790 0.69 PRCP (0.60) ACEHDAC8HDAC3HDAC1HDAC2
SCHEMBL15100399 0.69 PRCP (0.56) ACEOPRM1HDAC8HDAC3HDAC1
SCHEMBL14879190 0.69 PRCP (0.52) ACEOPRM1HDAC8HDAC3HDAC1
SCHEMBL12507462 0.68 PRCP (0.55) ACEOPRM1HDAC8HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed