SCHEMBL9744383

SCHEMBL9744383

CC(C)(C)NC(=O)C1c2ccccc2CCN1CC(O)CN1CCc2ccccc2C1C(=O)NC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 7/20 0.43
HDAC1 Q13547 6/20 0.43
HDAC3 O15379 5/20 0.43
NCOR2 Q9Y618 5/20 0.43
HDAC2 Q92769 4/20 0.43
TRPM8 Q7Z2W7 1/20 0.43
PRMT5 O14744 3/20 0.41
ACE P12821 1/20 0.41
OPRM1 P35372 1/20 0.41
WDR77 Q9BQA1 1/20 0.41
ACKR3 P25106 1/20 0.41
PRCP P42785 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40
KCNA5 P22460 1/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9012073 0.81 HDAC8 (0.42) HDAC8HDAC1HDAC3NCOR2HDAC2
SCHEMBL19960716 0.78 ACE (0.46) HDAC8HDAC1HDAC3NCOR2HDAC2
SCHEMBL18711701 0.78 TRPM8 (0.51) TRPM8ACEACKR3
SCHEMBL18711699 0.77 ACE (0.50) TRPM8ACEACKR3MEN1ALDH1A1
SCHEMBL18701726 0.77 TRPM8 (0.50) TRPM8ACEACKR3MEN1KMT2A
SCHEMBL18701727 0.77 TRPM8 (0.50) TRPM8ACEACKR3MEN1KMT2A
SCHEMBL18711706 0.75 RIPK1 (0.49) HDAC8TRPM8ACEACKR3MEN1
SCHEMBL8538945 0.73 CYP2C19 (0.52) HDAC8PRMT5ACEWDR77ALDH1A1
SCHEMBL3610720 0.72 XIAP (0.46) HDAC8HDAC1HDAC3NCOR2HDAC2
SCHEMBL3609137 0.69 ACE (0.52) HDAC8HDAC1HDAC3NCOR2HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed