SCHEMBL19960713

SCHEMBL19960713

NC(=O)C1c2ccccc2CCN1CC(F)F

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACE P12821 4/20 0.43
HDAC8 Q9BY41 5/20 0.41
F2RL1 P55085 1/20 0.41
HDAC3 O15379 4/20 0.40
NCOR2 Q9Y618 4/20 0.40
HDAC1 Q13547 3/20 0.40
HDAC2 Q92769 3/20 0.40
OPRM1 P35372 1/20 0.40
MTNR1B P49286 1/20 0.39
PRCP P42785 1/20 0.39
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19960716 0.83 ACE (0.46) ACEHDAC8HDAC3NCOR2HDAC1
SCHEMBL19960630 0.81 OPRM1 (0.43) ACEHDAC8HDAC1HDAC2OPRM1
SCHEMBL19953503 0.81 OPRM1 (0.43) ACEHDAC8HDAC1HDAC2OPRM1
SCHEMBL11472266 0.80 GRIN1 (0.50) ACEHDAC8HDAC3NCOR2HDAC1
SCHEMBL2848460 0.72 GRM2 (0.37) ACEHDAC8MTNR1B
SCHEMBL19960809 0.72 PRMT5 (0.42) ACEHDAC8F2RL1HDAC3NCOR2
SCHEMBL19960631 0.70 OPRM1 (0.38) ACEOPRM1MTNR1B
SCHEMBL16303966 0.69 ACE (0.50) ACEMTNR1BALDH1A1
SCHEMBL19960681 0.69 F11 (0.55) ACEF2RL1MTNR1BALDH1A1
SCHEMBL8293673 0.69 DPP4 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed