SCHEMBL19960809

SCHEMBL19960809

Cn1nccc1CN1CCc2ccccc2C1C(N)=O

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 1/20 0.42
WDR77 Q9BQA1 1/20 0.42
HDAC8 Q9BY41 9/20 0.40
HDAC1 Q13547 7/20 0.40
HDAC3 O15379 6/20 0.40
NCOR2 Q9Y618 6/20 0.40
HDAC2 Q92769 6/20 0.40
F2RL1 P55085 1/20 0.39
ACE P12821 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19960689 0.89 PRMT5 (0.40) PRMT5WDR77HDAC8HDAC1HDAC3
SCHEMBL19960810 0.87 PRMT5 (0.43) PRMT5WDR77HDAC8HDAC1HDAC3
SCHEMBL11472266 0.78 GRIN1 (0.50) HDAC8HDAC1HDAC3NCOR2HDAC2
SCHEMBL19960713 0.72 ACE (0.43) HDAC8HDAC1HDAC3NCOR2HDAC2
SCHEMBL6960867 0.70 PARP1 (0.36)
SCHEMBL6974370 0.69 XIAP (0.35)
SCHEMBL6970691 0.68 KDM4E (0.32) HDAC8HDAC1F2RL1
SCHEMBL6957978 0.68 SIRT1 (0.41)
SCHEMBL6966047 0.68 ESR1 (0.37) HDAC8HDAC1HDAC3NCOR2HDAC2
SCHEMBL23721558 0.67 KMT2A (0.41) PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed