SCHEMBL19971042

SCHEMBL19971042

COC(=O)C(N)CCc1ccc(O)c2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 6/20 0.43
LTA4H P09960 3/20 0.43
HDAC3 O15379 1/20 0.39
EP300 Q09472 1/20 0.39
KAT2B Q92831 1/20 0.39
KAT8 Q9H7Z6 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
MEN1 O00255 1/20 0.38
HCRTR1 O43613 1/20 0.38
KMT2A Q03164 1/20 0.38
KIF11 P52732 1/20 0.37
SLC2A1 P11166 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15804495 1.00 IDO1 (0.43) IDO1LTA4HHDAC3EP300KAT2B
SCHEMBL950509 0.85 IDO1 (0.46) IDO1LTA4HMEN1HCRTR1KMT2A
SCHEMBL15807803 0.85 IDO1 (0.46) IDO1LTA4HMEN1HCRTR1KMT2A
SCHEMBL15802471 0.84 KMT2A (0.46) IDO1LTA4HHDAC3EP300KAT2B
SCHEMBL20644869 0.83 MEN1 (0.41) IDO1MEN1HCRTR1KMT2ASLC2A1
Bromide SCHEMBL19971055 0.82 KMT2A (0.44) IDO1LTA4HHDAC3EP300KAT2B
Bromide SCHEMBL19971054 0.82 KMT2A (0.44) IDO1LTA4HHDAC3EP300KAT2B
SCHEMBL19983512 0.82 MEN1 (0.41) IDO1EP300MEN1HCRTR1KMT2A
SCHEMBL15802533 0.81 IDO1 (0.40) IDO1HDAC3EP300KAT2BKAT8
SCHEMBL9016080 0.80 MEN1 (0.57) MEN1HCRTR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2931712-B1 3,5-DIAMINO-6-CHLORO-N-(N-(4-PHENYLBUTYL)CARBAMIMIDOYL) PYRAZINE-2- CARBOXAMIDE COMPOUNDS PARION SCIENCES INC (US) 2018-03-21 EP disclosed