SCHEMBL19974449

SCHEMBL19974449

CC(C)(C)OC(=O)C1(c2cc(Cl)cc(CN3CCN(C(=O)OC(C(F)(F)F)C(F)(F)F)CC3)c2)CCCC1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 17/20 0.56
ABHD6 Q9BV23 8/20 0.56
PLA2G7 Q13093 6/20 0.56
CYP2D6 P10635 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19974356 0.88 MGLL (0.61) MGLLABHD6PLA2G7
SCHEMBL21082967 0.82 MGLL (0.63) MGLLABHD6PLA2G7CYP2D6
SCHEMBL28303847 0.80 DDR1 (0.40)
SCHEMBL19975519 0.80 CYP2D6 (0.51) MGLLCYP2D6
SCHEMBL18064816 0.80 MGLL (0.74) MGLLABHD6PLA2G7CYP2D6
SCHEMBL29532670 0.77 MGLL (0.61) MGLL
SCHEMBL20769556 0.77 MGLL (0.61) MGLL
SCHEMBL19974336 0.77 MGLL (0.67) MGLLABHD6PLA2G7CYP2D6
SCHEMBL19974335 0.76 MGLL (0.62) MGLLABHD6PLA2G7CYP2D6
SCHEMBL19974348 0.76 STS (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3515897-B1 PIPERAZINE CARBAMATES AS MODULATORS OF MAGL AND/OR ABHD6 AND THEIR USE H LUNDBECK AS (DK) 2021-08-18 EP disclosed
US-10899737-B2 Piperazine carbamates and methods of making and using same LUNDBECK LA JOLLA RESEARCH CENTER, INC. (US) 2021-01-26 US disclosed
EP-3515897-A1 PIPERAZINE CARBAMATES AND METHODS OF MAKING AND USING SAME Abide Therapeutics, Inc. (US) 2019-07-31 EP disclosed
US-20190202801-A1 PIPERAZINE CARBAMATES AND METHODS OF MAKING AND USING SAME H. LUNDBECK A/S (DK) 2019-07-04 US disclosed
WO-2018053447-A1 PIPERAZINE CARBAMATES AND METHODS OF MAKING AND USING SAME ABIDE THERAPEUTICS, INC. (US) 2018-03-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10899737-B2 Piperazine carbamates and methods of making and using same ABHD6, RABL6, ABHD16A MGLL 46/4885ABHD6 1/4885PLA2G7 204/4885
US-20190202801-A1 PIPERAZINE CARBAMATES AND METHODS OF MAKING AND USING SAME ABHD6, RABL6, ABHD16A MGLL 46/4885ABHD6 1/4885PLA2G7 204/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.