SCHEMBL19974692

SCHEMBL19974692

O=C(CCC1CCCC1)Oc1cnc[nH]1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 4/20 0.45
HTR3A P46098 1/20 0.45
MAPT P10636 1/20 0.43
HRH3 Q9Y5N1 3/20 0.43
ALDH1A1 P00352 1/20 0.43
IDO1 P14902 2/20 0.42
P2RX7 Q99572 2/20 0.42
HPGD P15428 2/20 0.42
MIF P14174 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19975547 0.74 HRH3 (0.43) HRH4HRH3
SCHEMBL19974772 0.73 KMT2A (0.43) HRH4HTR3AMAPTHRH3HPGD
SCHEMBL19974760 0.71 HRH3 (0.40) HRH4MAPTHRH3ALDH1A1IDO1
SCHEMBL19975114 0.70 HRH3 (0.42) HRH4MAPTHRH3ALDH1A1
SCHEMBL15059972 0.70 EPHX1 (0.50) HRH4HRH3ALDH1A1
SCHEMBL19974645 0.69 MEN1 (0.38) MAPTHRH3ALDH1A1
SCHEMBL28006498 0.68 KLK7 (0.56) ALDH1A1HPGD
SCHEMBL27673261 0.68 HRH4 (0.36) HRH4MAPTHRH3ALDH1A1
SCHEMBL30799954 0.68 HPGD (0.48) MAPTHPGD
SCHEMBL21396239 0.67 KLK7 (0.51) MAPTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512840-A1 NOVEL SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS D-AMINO ACID OXIDASE (DAAO) INHIBITORS Tseng, Yufeng, Jane (US) 2019-07-24 EP disclosed
WO-2018053161-A1 NOVEL SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS D-AMINO ACID OXIDASE (DAAO) INHIBITORS NATIONAL TAIWAN UNIVERSITY (TW) 2018-03-22 WO disclosed