SCHEMBL19976489

SCHEMBL19976489

Nc1ccc(C(=O)NCCC(F)(F)F)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.54
MAPT P10636 1/20 0.54
HIF1A Q16665 1/20 0.54
SLC22A6 Q4U2R8 1/20 0.54
SLC22A8 Q8TCC7 1/20 0.54
LMNA P02545 3/20 0.54
MLYCD O95822 3/20 0.54
TSHR P16473 2/20 0.54
SLC22A2 O15244 1/20 0.54
SLC22A1 O15245 1/20 0.54
ALDH1A1 P00352 1/20 0.54
ACHE P22303 1/20 0.54
MAPK1 P28482 1/20 0.54
CYP2C19 P33261 1/20 0.54
ESRRG P62508 1/20 0.54
BLM P54132 1/20 0.53
PMP22 Q01453 1/20 0.53
HDAC3 O15379 4/20 0.51
HDAC4 P56524 3/20 0.51
HDAC1 Q13547 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23222129 0.90 HDAC3 (0.52) KDM4EMAPTHIF1ASLC22A6SLC22A8
SCHEMBL16964203 0.86 MLYCD (0.54) MLYCDTSHRALDH1A1BLMPMP22
SCHEMBL16964231 0.84 MLYCD (0.55) LMNAMLYCDALDH1A1MAPK1HDAC3
SCHEMBL507116 0.83 HDAC3 (0.54) MLYCDTSHRALDH1A1ESRRGBLM
SCHEMBL9344489 0.83 KDM4E (0.68) KDM4EMAPTHIF1ASLC22A6SLC22A8
SCHEMBL16964142 0.83 MLYCD (0.54) MLYCDHDAC3CYP1A2
SCHEMBL19938019 0.83 MLYCD (0.67) KDM4EMAPTHIF1ASLC22A6SLC22A8
SCHEMBL16964303 0.83 MLYCD (0.58) LMNAMLYCDALDH1A1MAPK1HDAC3
SCHEMBL18359001 0.83 LMNA (0.62) LMNAMLYCDALDH1A1HDAC3POLB
SCHEMBL8507100 0.82 HDAC3 (0.62) LMNAMLYCDESRRGHDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9920042-B2 Compounds for use in the treatment of mycobacterial infections UNIVERSITE DE DROIT ET DE LA SANTE DE LILLE 2 (FR) 2018-03-20 US disclosed