SCHEMBL19976852

SCHEMBL19976852

CC(C)(C)N/C(=N/C(=O)c1ccc(C(F)(F)F)cc1)Nc1n[nH]c2ncccc12

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.40
TRPV1 Q8NER1 10/20 0.39
CRHR1 P34998 1/20 0.39
RIPK1 Q13546 1/20 0.38
GSK3B P49841 2/20 0.38
MAPK10 P53779 1/20 0.37
TLR7 Q9NYK1 1/20 0.36
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19976929 0.85 RIPK1 (0.37) HDAC6TRPV1RIPK1AURKAAURKB
SCHEMBL18558644 0.79 TRPV1 (0.38) HDAC6TRPV1GSK3B
SCHEMBL9920889 0.76 HDAC6 (0.37) HDAC6TRPV1GSK3B
SCHEMBL9921034 0.74 HDAC6 (0.39) HDAC6TRPV1GSK3BTLR7
SCHEMBL18558594 0.74 HDAC6 (0.39) HDAC6TRPV1GSK3B
SCHEMBL19976725 0.74 GSK3B (0.52) HDAC6GSK3BMAPK10
SCHEMBL19976736 0.74 MAP2K4 (0.44) HDAC6GSK3BMAPK10AURKAAURKB
SCHEMBL18558030 0.73 GRM5 (0.41) TRPV1GSK3BAURKB
SCHEMBL9905332 0.73 P2RY14 (0.38) HDAC6TRPV1TLR7
SCHEMBL9905327 0.73 P2RY14 (0.38) HDAC6TRPV1TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9920012-B2 Indazole guanidine F1F0-ATPase inhibitors and therapeutic uses thereof LYCERA CORPORATION (US) 2018-03-20 US disclosed