SCHEMBL19978884

SCHEMBL19978884

COc1nc(F)nc2[nH]cnc12

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.36
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
BRD4 O60885 1/20 0.31
ABL1 P00519 1/20 0.31
RAD52 P43351 1/20 0.31
RIN1 Q13671 1/20 0.31
DYRK1A Q13627 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31380770 0.79 XDH (0.37) PDPK1CYP1A2CYP2C19ABL1RAD52
Methylguanine SCHEMBL1336757 0.79 CDK1 (0.41) PDPK1
SCHEMBL22700363 0.79 MEN1 (0.37) PDPK1CYP1A2CYP2C19ABL1RAD52
SCHEMBL9503831 0.79 PDPK1 (0.36) PDPK1CYP1A2CYP2C19ABL1RAD52
SCHEMBL1443986 0.79 XDH (0.37) PDPK1CYP1A2CYP2C19ABL1RAD52
SCHEMBL4525138 0.78 HPGD (0.35) PDPK1CYP1A2CYP2C19
SCHEMBL18961720 0.76 GAA (0.35) PDPK1CYP1A2CYP2C19
SCHEMBL9925954 0.76 PDPK1 (0.34) PDPK1DYRK1A
SCHEMBL2526551 0.75 PARP1 (0.32) PDPK1DYRK1A
SCHEMBL8959020 0.73 MGMT (0.46) CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512860-B1 NUCLEOSIDE AND NUCLEOTIDE ANALOGUES BEARING A QUATERNARY ALL-CARBON STEREOGENIC CENTER AT THE 2' POSITION AND METHODS OF USE AS A CARDIOPROTECTIVE AGENT LCB PHARMA INC (CA) 2020-11-25 EP disclosed
WO-2018049534-A1 NUCLEOSIDE AND NUCLEOTIDE ANALOGUES BEARING A QUATERNARY ALL-CARBON STEREOGENIC CENTER AT THE 2' POSITION AND METHODS OF USE AS A CARDIOPROTECTIVE AGENT LCB PHARMA INC. (CA) 2018-03-22 WO disclosed