SCHEMBL19980649

SCHEMBL19980649

CC(C)(C#N)c1ccc(C=O)cc1NC=O

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ALDH1A1 P00352 2/20 0.32
TSHR P16473 1/20 0.32
EGFR P00533 1/20 0.32
KDM4E B2RXH2 1/20 0.31
PTGS2 P35354 1/20 0.31
RAB9A P51151 1/20 0.31
KIF11 P52732 1/20 0.30
CYP2A6 P11509 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19980704 0.78 MAPT (0.34) MAPTMAPK1NPSR1
SCHEMBL309292 0.78 KIF11 (0.45) ALDH1A1TSHREGFRKDM4EPTGS2
SCHEMBL25135200 0.76 KDM4E (0.44) MAPTALDH1A1KDM4ERAB9AKIF11
SCHEMBL22298702 0.69 ALDH1A1 (0.37) MAPTALDH1A1TSHRKDM4EPTGS2
SCHEMBL472590 0.69 EGFR (0.44) NPSR1ALDH1A1EGFRKDM4ECYP2A6
SCHEMBL31270677 0.67 KDM5A (0.58) MAPTMAPK1ALDH1A1TSHREGFR
SCHEMBL2517047 0.67 ALDH1A1 (0.41) ALDH1A1RAB9ACYP2A6
SCHEMBL8067987 0.65 CYP19A1 (0.38) EGFR
SCHEMBL11328597 0.64 ALDH1A1 (0.42) NPSR1ALDH1A1TSHRKDM4EPTGS2
SCHEMBL393655 0.64 MAPT (0.40) MAPTMAPK1NPSR1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512850-B1 INHIBITORS OF THE MENIN-MLL INTERACTION VITAE PHARMACEUTICALS LLC (US) 2023-04-12 EP disclosed
WO-2018053267-A1 INHIBITORS OF THE MENIN-MLL INTERACTION VITAE PHARMACEUTICALS, INC. (US) 2018-03-22 WO disclosed