SCHEMBL19981613

SCHEMBL19981613

O=S(=O)(Oc1ccc2c(c1)CNCC2)C(F)(F)F

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PNMT P11086 9/20 0.51
ADRA2A P08913 2/20 0.51
ADRA2B P18089 2/20 0.51
ADRA2C P18825 2/20 0.51
HTR2C P28335 1/20 0.46
HTR7 P34969 1/20 0.46
HTR6 P50406 1/20 0.46
DRD2 P14416 1/20 0.45
HTR1D P28221 1/20 0.45
DRD3 P35462 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14302335 0.94 ASIC3 (0.46) PNMTADRA2AADRA2BADRA2CHTR2C
Hydrochloric Acid SCHEMBL17965626 0.93 ASIC3 (0.45) PNMTADRA2AADRA2BADRA2CHTR2C
SCHEMBL28451134 0.87 HTR1D (0.43) HTR2CHTR7HTR6DRD2HTR1D
SCHEMBL6979583 0.80 PNMT (0.50) PNMTADRA2AADRA2BADRA2CDRD2
SCHEMBL7443640 0.79 DRD2 (0.44) HTR2CHTR7HTR6DRD2HTR1D
SCHEMBL5026108 0.79 STS (0.64) HTR2CHTR7HTR6DRD2HTR1D
SCHEMBL4427945 0.79 STS (0.59) DRD2HTR1DDRD3
SCHEMBL29051886 0.78 DRD2 (0.43) HTR2CHTR7HTR6DRD2HTR1D
Hydrochloric Acid SCHEMBL15422486 0.78 PNMT (0.49) PNMTADRA2AADRA2BADRA2CDRD2
SCHEMBL17921501 0.78 PNMT (0.61) PNMTADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053222-A1 TETRAHYDROISOQUINOLINE KAPPA OPIOID ANTAGONISTS RESEARCH TRAINGLE INSTITUTE (US) 2018-03-22 WO disclosed