SCHEMBL19982177

SCHEMBL19982177

COC(=O)C(Cc1ccccc1)NC(=O)CC1CCN(C(=O)C2CCCN2C)CC1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
YAP1 P46937 14/20 0.60
GAA P10253 1/20 0.54
IL2RA P01589 1/20 0.53
ALB P02768 1/20 0.53
IL2 P60568 1/20 0.53
ATM Q13315 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19982079 0.93 YAP1 (0.73) YAP1GAAIL2RAALBIL2
SCHEMBL19982077 0.92 YAP1 (0.55) YAP1GAAIL2RAALBIL2
SCHEMBL19982179 0.90 YAP1 (0.59) YAP1GAAIL2RAALBIL2
SCHEMBL19976384 0.85 YAP1 (0.69) YAP1GAAIL2RAALBIL2
SCHEMBL19976383 0.85 YAP1 (0.69) YAP1GAAIL2RAALBIL2
SCHEMBL19982078 0.83 YAP1 (0.72) YAP1IL2RAALBIL2
SCHEMBL27389203 0.82 GAA (0.58) GAAATML3MBTL1CYP3A4CYP2D6
SCHEMBL19982076 0.81 YAP1 (0.54) YAP1IL2RAALBIL2
SCHEMBL19975557 0.81 YAP1 (0.54) YAP1
SCHEMBL19982213 0.80 YAP1 (0.85) YAP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053446-A1 YAP1 INHIBITORS THAT TARGET THE INTERACTION OF YAP1 WITH OCT4 H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2018-03-22 WO disclosed