SCHEMBL19982678

SCHEMBL19982678

CC(=O)c1ccc2nc(-c3ccccc3)[nH]c2c1

nearest known ligand 0.74

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 10/20 0.74
HDAC3 O15379 1/20 0.67
HDAC1 Q13547 1/20 0.67
HDAC8 Q9BY41 1/20 0.67
HDAC6 Q9UBN7 1/20 0.67
PLAU P00749 1/20 0.66
PRSS1 P07477 1/20 0.66
NPBWR1 P48145 2/20 0.61
NR4A2 P43354 1/20 0.60
MEN1 O00255 1/20 0.60
KMT2A Q03164 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6450749 0.91 NPBWR1 (0.71) CHEK2HDAC3HDAC1HDAC8HDAC6
SCHEMBL27765862 0.88 CHEK2 (0.78) CHEK2HDAC3HDAC1HDAC8HDAC6
SCHEMBL3178116 0.88 CHEK2 (0.78) CHEK2HDAC3HDAC1HDAC8HDAC6
SCHEMBL19753931 0.86 CHEK2 (0.67) CHEK2NPBWR1NR4A2MEN1KMT2A
SCHEMBL2243148 0.85 CHEK2 (0.80) CHEK2HDAC3HDAC1HDAC8HDAC6
SCHEMBL2649653 0.85 HDAC6 (0.76) CHEK2HDAC3HDAC1HDAC8HDAC6
SCHEMBL2617479 0.85 KDM4E (0.71) CHEK2HDAC3HDAC1HDAC8HDAC6
SCHEMBL18237054 0.83 HDAC6 (0.95) CHEK2HDAC3HDAC1HDAC8HDAC6
SCHEMBL19986735 0.82 CYP1A2 (0.59) CHEK2HDAC3HDAC1HDAC8HDAC6
SCHEMBL13808897 0.82 HDAC6 (0.74) CHEK2HDAC3HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018050771-A1 BENZIMIDAZOL DERIVATIVES FOR TREATING FILOVIRUS INFECTION CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2018-03-22 WO disclosed