SCHEMBL19983057

SCHEMBL19983057

CC(C)(C)OC(=O)NCCCC[C@@H](NC(=O)c1cccc(N=[N+]=N)c1)C(=O)COc1c(F)cccc1F

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSH P09668 1/20 0.41
CTSK P43235 1/20 0.41
TDP1 Q9NUW8 3/20 0.40
PAX8 Q06710 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19983008 0.92 CTSH (0.41) CTSHCTSKTDP1PAX8KDM4E
SCHEMBL19983290 0.92 CTSH (0.41) CTSHCTSKTDP1PAX8KDM4E
SCHEMBL19983223 0.89 CTSH (0.42) CTSHCTSKTDP1PAX8KDM4E
SCHEMBL19983222 0.88 CA1 (0.42) TDP1PAX8KDM4EMAPTNPSR1
SCHEMBL19983025 0.87 CTSH (0.46) CTSHCTSKTDP1PAX8KDM4E
SCHEMBL17646256 0.86 CTSK (0.40) CTSHCTSKTDP1KDM4EMAPT
SCHEMBL19665687 0.86 CTSK (0.40) CTSHCTSKTDP1KDM4EMAPT
SCHEMBL19983306 0.85 TDP1 (0.46) TDP1PAX8KDM4EMAPTNPSR1
SCHEMBL19982961 0.84 CTSK (0.44) CTSHCTSKTDP1PAX8
SCHEMBL19983003 0.84 CTSK (0.44) CTSHCTSKTDP1PAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053353-A1 KETONE INHIBITORS OF LYSINE GINGIPAIN Cortexyme, Inc. (US) 2018-03-22 WO disclosed