SCHEMBL19983082

SCHEMBL19983082

CC1=CC(C)=[N+]2C1=Cc1ccc(CCC(=O)NCc3cn(-c4cccc(C(N)=O)c4)nn3)n1S2(F)F

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP14 Q460N5 1/20 0.39
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
ALK Q9UM73 2/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
MIF P14174 1/20 0.33
NOTUM Q6P988 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
RXRA P19793 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
TYMS P04818 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16238217 0.60 MAOA (0.54) MAOAMAOBALKMIFNOTUM
SCHEMBL29300000 0.56 NOTUM (0.66) MAOACA1CA2MIFNOTUM
SCHEMBL16785620 0.56 CA2 (0.62) CA12CA1CA2CA9NOTUM
SCHEMBL16250023 0.55 CA1 (0.64) MAOAMAOBALKCA12CA1
SCHEMBL27423391 0.54 KDM1A (0.54) CA12CA1CA2CA9NOTUM
SCHEMBL19365353 0.54 CA1 (0.60) CA12CA1CA2CA9NOTUM
SCHEMBL4583569 0.54 TP53 (0.70) NOTUM
SCHEMBL29299489 0.53 MIF (0.58) MAOAMIFNOTUM
SCHEMBL27430548 0.53 CA1 (0.58) CA12CA1CA2CA9RXRA
SCHEMBL22416987 0.53 MAOA (0.46) PARP14MAOAMAOBCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053353-A1 KETONE INHIBITORS OF LYSINE GINGIPAIN Cortexyme, Inc. (US) 2018-03-22 WO disclosed