SCHEMBL19984341

SCHEMBL19984341

CO[C@H]1CC[C@H](O[Si](c2ccccc2)(c2ccccc2)C(C)(C)C)CC1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.40
DPP4 P27487 1/20 0.36
ADORA3 P0DMS8 1/20 0.33
MAPK8 P45983 1/20 0.32
MAPK10 P53779 1/20 0.32
MAPK1 P28482 1/20 0.31
GBA1 P04062 1/20 0.31
CYP3A4 P08684 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
SMYD2 Q9NRG4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14461324 0.93 BACE1 (0.43) BACE1MAPK1CYP3A4HTTSMN1; SMN2
SCHEMBL25417788 0.87 BACE1 (0.36) BACE1DPP4CYP3A4HTTSMN1; SMN2
SCHEMBL29498916 0.86 BACE1 (0.42) BACE1CYP3A4HTTSMN1; SMN2SMYD2
SCHEMBL359522 0.85 BACE1 (0.40) BACE1CYP3A4HTTSMN1; SMN2SMYD2
SCHEMBL14630717 0.85 BACE1 (0.40) BACE1CYP3A4HTTSMN1; SMN2SMYD2
SCHEMBL14630715 0.85 BACE1 (0.40) BACE1CYP3A4HTTSMN1; SMN2SMYD2
SCHEMBL4797973 0.85 BACE1 (0.40) BACE1CYP3A4HTTSMN1; SMN2SMYD2
SCHEMBL241741 0.85 BACE1 (0.40) BACE1CYP3A4HTTSMN1; SMN2SMYD2
SCHEMBL14840794 0.85 BACE1 (0.40) BACE1CYP3A4HTTSMN1; SMN2SMYD2
SCHEMBL26663762 0.85 BACE1 (0.40) BACE1CYP3A4HTTSMN1; SMN2SMYD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10233156-B2 9-membered fused ring derivative SHIONOGI & CO., LTD. (JP) 2019-03-19 US disclosed
US-20180079727-A1 9-MEMBERED FUSED RING DERIVATIVE SHIONOGI & CO., LTD. (JP) 2018-03-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180079727-A1 9-MEMBERED FUSED RING DERIVATIVE ACSS2, AGTR2, ACSL3 BACE1 1435/4885DPP4 3206/4885ADORA3 763/4885
US-10233156-B2 9-membered fused ring derivative AGTR2, ACSS2, ACSL3 BACE1 1632/4885DPP4 2869/4885ADORA3 673/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.