SCHEMBL19986373

SCHEMBL19986373

CCc1cn(C(C)C(=O)O)nn1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 6/20 0.40
MAPK14 Q16539 2/20 0.36
LGALS3 P17931 1/20 0.34
PTPN1 P18031 1/20 0.34
CDC25B P30305 1/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
GLA P06280 1/20 0.33
HTT P42858 1/20 0.33
ATM Q13315 1/20 0.33
GPR88 Q9GZN0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5998647 0.86 NOTUM (0.41) CYP19A1MAPK14LGALS3
SCHEMBL24878799 0.79 CYP19A1 (0.40) CYP19A1MAPK14POLB
SCHEMBL22854013 0.77 CYP19A1 (0.39) CYP19A1POLB
SCHEMBL908039 0.77 ALDH1A1 (0.41) MAPK14ALDH1A1POLBHTTATM
SCHEMBL24878496 0.76 CYP19A1 (0.39) CYP19A1MAPK14POLB
SCHEMBL22854014 0.75 CYP19A1 (0.38) CYP19A1POLBHTTATM
SCHEMBL13872394 0.75 ALDH1A1 (0.40) MAPK14ALDH1A1HTTATM
SCHEMBL20926022 0.74 CYP19A1 (0.40) CYP19A1POLB
SCHEMBL19901549 0.74 CYP19A1 (0.44) CYP19A1POLB
SCHEMBL24974351 0.74 CYP19A1 (0.40) CYP19A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053517-A1 INHIBITORS OF LDLR-PCSK9 PROTEIN-PROTEIN INTERACTION AND METHODS OF THEIR USE THE TEXAS A&M UNIVERSITY SYSTEM (US) 2018-03-22 WO disclosed