SCHEMBL19986502

SCHEMBL19986502

O=C(NCCCNc1c(Cl)cncc1Cl)Nc1ccc(F)c(Cl)c1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.60
MEN1 O00255 6/20 0.60
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C19 P33261 1/20 0.53
LMNA P02545 4/20 0.53
MAPT P10636 1/20 0.53
HTT P42858 3/20 0.52
TP53 P04637 1/20 0.52
SLC2A1 P11166 1/20 0.51
NPC1 O15118 2/20 0.50
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
ALOX15 P16050 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
EPHX2 P34913 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986566 0.93 MEN1 (0.51) KMT2AMEN1CYP1A2CYP3A4CYP2C19
SCHEMBL19986553 0.93 KMT2A (0.63) KMT2AMEN1CYP1A2CYP3A4CYP2C19
SCHEMBL19986669 0.91 MEN1 (0.48) KMT2AMEN1CYP1A2CYP3A4CYP2C19
SCHEMBL19986530 0.89 ALOX15 (0.58) KMT2AMEN1LMNAMAPTHTT
SCHEMBL19986578 0.86 MEN1 (0.41) KMT2AMEN1CYP1A2CYP3A4CYP2C19
SCHEMBL19986563 0.86 MEN1 (0.53) KMT2AMEN1CYP1A2CYP3A4CYP2C19
SCHEMBL19986701 0.85 MARS1 (0.59) KMT2AMEN1LMNAHTTTP53
SCHEMBL19986568 0.85 EPHX1 (0.60) KMT2AMEN1CYP1A2CYP3A4CYP2C19
SCHEMBL19986714 0.84 ALOX15 (0.43) KMT2AMEN1CYP1A2CYP3A4CYP2C19
SCHEMBL19986712 0.84 MEN1 (0.47) KMT2AMEN1LMNAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429341-A Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-09-24 CN disclosed
CN-109790123-B Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-06-25 CN disclosed
WO-2018050110-A1 NOVEL CAPSID PROTEIN ASSEMBLY INHIBITOR 正大天晴药业集团股份有限公司 2018-03-22 WO disclosed