SCHEMBL19986578

SCHEMBL19986578

O=C(NCCCNc1c(Cl)cncc1Cl)Nc1cc(F)c(F)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
CDK2 P24941 1/20 0.39
FLT4 P35916 1/20 0.39
MARS1 P56192 2/20 0.38
ALOX15 P16050 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C19 P33261 2/20 0.38
CNR1 P21554 3/20 0.38
EPHX2 P34913 1/20 0.37
SLC6A3 Q01959 2/20 0.36
EPHX1 P07099 3/20 0.36
LMNA P02545 2/20 0.36
NAMPT P43490 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986506 0.93 MEN1 (0.43) MEN1KMT2AALOX15HSD17B10CYP1A2
SCHEMBL19986566 0.88 MEN1 (0.51) MEN1KMT2AMARS1ALOX15HSD17B10
SCHEMBL19986669 0.88 MEN1 (0.48) MEN1KMT2AMARS1ALOX15HSD17B10
SCHEMBL19986712 0.86 MEN1 (0.47) MEN1KMT2ACDK2FLT4MARS1
SCHEMBL19986714 0.86 ALOX15 (0.43) MEN1KMT2ACDK2FLT4MARS1
SCHEMBL19986705 0.86 MARS1 (0.47) MEN1KMT2AMARS1ALOX15HSD17B10
SCHEMBL19986502 0.86 KMT2A (0.60) MEN1KMT2AALOX15HSD17B10CYP1A2
SCHEMBL19986701 0.82 MARS1 (0.59) MEN1KMT2ACDK2FLT4MARS1
SCHEMBL19986530 0.81 ALOX15 (0.58) MEN1KMT2AALOX15HSD17B10EPHX2
SCHEMBL19986671 0.81 EPHX2 (0.49) MEN1KMT2AALOX15HSD17B10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429341-A Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-09-24 CN disclosed
CN-109790123-B Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-06-25 CN disclosed
WO-2018050110-A1 NOVEL CAPSID PROTEIN ASSEMBLY INHIBITOR 正大天晴药业集团股份有限公司 2018-03-22 WO disclosed