SCHEMBL19986540

SCHEMBL19986540

COC(CNC(=O)Nc1cccc(Cl)c1)CNc1c(Cl)cncc1Cl

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.47
NPC1 O15118 2/20 0.47
EPHX1 P07099 4/20 0.46
OPRM1 P35372 1/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
LMNA P02545 2/20 0.45
MAPT P10636 2/20 0.45
HTT P42858 2/20 0.45
ALDH1A1 P00352 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
EPHX2 P34913 2/20 0.44
CASR P41180 1/20 0.44
POLB P06746 1/20 0.44
TRPV1 Q8NER1 1/20 0.43
MTOR P42345 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986723 0.89 MEN1 (0.42) MEN1KMT2ALMNAMAPTALDH1A1
SCHEMBL19986697 0.87 RAB9A (0.47) RAB9ANPC1EPHX1OPRM1MEN1
SCHEMBL19986539 0.87 LMNA (0.58) RAB9ANPC1MEN1KMT2ALMNA
SCHEMBL19986666 0.85 LMNA (0.39) RAB9AMEN1KMT2ALMNAMAPT
SCHEMBL19986622 0.85 NPC1 (0.51) RAB9ANPC1EPHX1OPRM1MEN1
SCHEMBL19986628 0.80 MEN1 (0.56) RAB9ANPC1EPHX1MEN1KMT2A
SCHEMBL19986568 0.78 EPHX1 (0.60) RAB9ANPC1EPHX1MEN1KMT2A
SCHEMBL19986717 0.74 MEN1 (0.44) RAB9AMEN1KMT2ALMNAMAPT
SCHEMBL19986623 0.73 MEN1 (0.45) RAB9AMEN1KMT2ALMNAMAPT
SCHEMBL19986611 0.73 LMNA (0.50) RAB9ANPC1EPHX1OPRM1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429341-A Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-09-24 CN disclosed
CN-109790123-B Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-06-25 CN disclosed
WO-2018050110-A1 NOVEL CAPSID PROTEIN ASSEMBLY INHIBITOR 正大天晴药业集团股份有限公司 2018-03-22 WO disclosed