SCHEMBL19986697

SCHEMBL19986697

COC(CNC(=O)Nc1ccc(Cl)c(Cl)c1)CNc1c(Cl)cncc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.47
ALDH1A1 P00352 1/20 0.46
EPHX1 P07099 2/20 0.45
EPHX2 P34913 2/20 0.45
LMNA P02545 3/20 0.45
OPRL1 P41146 1/20 0.44
NPC1 O15118 7/20 0.43
HPGD P15428 2/20 0.43
MAPK1 P28482 1/20 0.43
MAPT P10636 4/20 0.42
HTT P42858 2/20 0.42
GLA P06280 1/20 0.42
KMT2A Q03164 6/20 0.42
MEN1 O00255 5/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP2D6 P10635 1/20 0.42
CA2 P00918 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986539 0.91 LMNA (0.58) RAB9AALDH1A1LMNANPC1MAPT
SCHEMBL19986666 0.89 LMNA (0.39) RAB9AALDH1A1LMNAOPRL1MAPT
SCHEMBL19986540 0.87 RAB9A (0.47) RAB9AALDH1A1EPHX1EPHX2LMNA
SCHEMBL19986723 0.87 MEN1 (0.42) ALDH1A1LMNAMAPTKMT2AMEN1
SCHEMBL19986611 0.85 LMNA (0.50) RAB9AALDH1A1EPHX1EPHX2LMNA
SCHEMBL19986475 0.84 RAB9A (0.50) RAB9AALDH1A1EPHX1EPHX2LMNA
SCHEMBL19986530 0.77 ALOX15 (0.58) RAB9AALDH1A1EPHX1EPHX2LMNA
SCHEMBL19986720 0.76 RAB9A (0.49) RAB9AALDH1A1EPHX1EPHX2LMNA
SCHEMBL19986510 0.76 LMNA (0.65) RAB9AALDH1A1LMNANPC1MAPT
SCHEMBL19986463 0.75 LMNA (0.60) RAB9AALDH1A1LMNANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429341-A Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-09-24 CN disclosed
CN-109790123-B Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-06-25 CN disclosed
WO-2018050110-A1 NOVEL CAPSID PROTEIN ASSEMBLY INHIBITOR 正大天晴药业集团股份有限公司 2018-03-22 WO disclosed