SCHEMBL19986732

SCHEMBL19986732

C/C(=C\C=C(/C)C(F)(F)F)NC(=O)N1CCN(Cc2ccc3nc(-c4ccccc4)[nH]c3c2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 3/20 0.48
BCHE P06276 2/20 0.46
ACHE P22303 2/20 0.46
HDAC6 Q9UBN7 4/20 0.46
HDAC3 O15379 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
HTR1A P08908 1/20 0.45
DRD2 P14416 1/20 0.45
HTR2A P28223 1/20 0.45
AURKA O14965 3/20 0.42
CDK1 P06493 3/20 0.42
CCNB1 P14635 3/20 0.42
CDK2 P24941 3/20 0.42
AURKB Q96GD4 3/20 0.42
FGFR1 P11362 2/20 0.42
FLT1 P17948 1/20 0.42
FAAH O00519 1/20 0.41
CHEK2 O96017 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986738 0.92 SLC2A1 (0.46) SLC2A1HDAC6HDAC3HDAC1HDAC2
SCHEMBL19970728 0.78 FAAH (0.63) SLC2A1AURKACDK1CCNB1CDK2
SCHEMBL19970873 0.77 FAAH (0.61) AURKACDK1CCNB1CDK2AURKB
SCHEMBL19970828 0.74 NPBWR1 (0.64) SLC2A1BCHEACHEHDAC6HDAC3
SCHEMBL19970835 0.73 BCHE (0.53) SLC2A1BCHEACHEHDAC6HDAC3
SCHEMBL19970807 0.72 ACACB (0.62) SLC2A1BCHEACHEHDAC6HDAC3
SCHEMBL19970727 0.72 FAAH (0.63) SLC2A1FAAH
SCHEMBL19970741 0.71 RUNX1 (0.61) SLC2A1BCHEACHEHTR1ADRD2
SCHEMBL19970777 0.71 SLC2A1 (0.58) SLC2A1BCHEACHEHDAC6HDAC3
SCHEMBL19970830 0.70 FAAH (0.56) SLC2A1AURKACDK1CCNB1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3296297-A1 BENZIMIDAZOL DERIVATIVES FOR TREATING FILOVIRUS INFECTION CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2018-03-21 EP disclosed