SCHEMBL19986738

SCHEMBL19986738

C/C(=C\C=C(/C)C(F)(F)F)NC(=O)N1CCN(Cc2ccc3nc(-c4cccnc4)[nH]c3c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 2/20 0.46
ALDH1A1 P00352 3/20 0.45
HPGD P15428 2/20 0.45
HSD17B10 Q99714 1/20 0.45
AURKA O14965 1/20 0.44
CDK1 P06493 1/20 0.44
CCNB1 P14635 1/20 0.44
CDK2 P24941 1/20 0.44
AURKB Q96GD4 1/20 0.44
KIT P10721 7/20 0.42
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
TP53 P04637 3/20 0.41
KDM4E B2RXH2 2/20 0.41
TBK1 Q9UHD2 1/20 0.40
CYP11B1 P15538 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986732 0.92 SLC2A1 (0.48) SLC2A1AURKACDK1CCNB1CDK2
SCHEMBL19970830 0.80 FAAH (0.56) SLC2A1ALDH1A1HPGDHSD17B10AURKA
SCHEMBL19970868 0.79 ALDH1A1 (0.55) ALDH1A1HPGDHSD17B10AURKACDK1
SCHEMBL19970798 0.76 KCNH2 (0.62) SLC2A1ALDH1A1HPGDAURKACDK1
SCHEMBL19970737 0.74 SLC2A1 (0.57) SLC2A1KITHDAC3HDAC1HDAC2
SCHEMBL19970829 0.74 FAAH (0.56) SLC2A1KITFAAH
SCHEMBL19970730 0.74 RUNX1 (0.54) SLC2A1ALDH1A1HPGDAURKACDK1
SCHEMBL19970764 0.74 AURKA (0.47) SLC2A1ALDH1A1HPGDHSD17B10AURKA
SCHEMBL19970867 0.73 FAAH (0.54) ALDH1A1HPGDHSD17B10KITFAAH
SCHEMBL19970841 0.72 RUNX1 (0.53) SLC2A1ALDH1A1HPGDAURKACDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3296297-A1 BENZIMIDAZOL DERIVATIVES FOR TREATING FILOVIRUS INFECTION CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2018-03-21 EP disclosed