SCHEMBL19987417

SCHEMBL19987417

Cc1ccc2c(c1)C1(c3cc(C)ccc3-2)c2cc(C)ccc2-c2ccc(N3c4ccccc4C(C)(c4ccccc4)c4ccccc43)cc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 2/20 0.36
PGR P06401 1/20 0.34
ALDH1A1 P00352 3/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
PAX8 Q06710 1/20 0.33
MCL1 Q07820 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAPT P10636 1/20 0.33
KDM4E B2RXH2 2/20 0.33
HSD17B10 Q99714 1/20 0.33
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CRHBP P24387 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
ATM Q13315 1/20 0.31
CRHR2 Q13324 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19987411 0.97 PDK2 (0.37) PDK2PGRALDH1A1LMNAGAA
SCHEMBL15183660 0.90 PDK2 (0.38) PDK2PGRALDH1A1LMNAMAPT
SCHEMBL808059 0.88 PGR (0.40) PDK2PGRALDH1A1LMNAL3MBTL1
SCHEMBL15183636 0.87 PDK2 (0.39) PDK2PGRALDH1A1LMNAMAPT
SCHEMBL15627514 0.86 PDK2 (0.36) PDK2PGRALDH1A1LMNAGAA
SCHEMBL15627532 0.86 PDK2 (0.37) PDK2PGRALDH1A1LMNAGAA
SCHEMBL15183634 0.85 PGR (0.42) PDK2PGRALDH1A1KDM4EHSD17B10
SCHEMBL17901851 0.84 PDK2 (0.37) PDK2PGRALDH1A1LMNAGAA
SCHEMBL20842752 0.84 ITGB2 (0.33) ALDH1A1LMNAGAAPAX8MCL1
SCHEMBL17901883 0.84 PDK2 (0.39) PDK2ALDH1A1LMNAGAAPAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2826079-B1 ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2021-01-20 EP disclosed
EP-2907173-B1 ELECTRONIC DEVICE MERCK PATENT GMBH (DE) 2018-03-21 EP disclosed