SCHEMBL19987464

SCHEMBL19987464

CCCC(C)c1ccc(Cl)cc1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
HTT P42858 1/20 0.39
KCNH2 Q12809 1/20 0.37
CXCR3 P49682 1/20 0.35
MDM2 Q00987 1/20 0.35
PSEN1 P49768 3/20 0.34
PSEN2 P49810 3/20 0.34
APH1B Q8WW43 3/20 0.34
NCSTN Q92542 3/20 0.34
APH1A Q96BI3 3/20 0.34
PSENEN Q9NZ42 3/20 0.34
DPP4 P27487 1/20 0.34
DPP7 Q9UHL4 1/20 0.34
SLC6A4 P31645 1/20 0.34
PPARG P37231 3/20 0.33
PPARA Q07869 3/20 0.33
PNMT P11086 1/20 0.33
OPRM1 P35372 1/20 0.33
S1PR1 P21453 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19464670 0.88 MAPT (0.38) LMNATP53HTTKCNH2CXCR3
SCHEMBL22932512 0.87 PSEN1 (0.37) LMNATP53HTTPSEN1PSEN2
SCHEMBL19121860 0.85 LMNA (0.41) LMNATP53HTTKCNH2CXCR3
SCHEMBL16117013 0.85 LMNA (0.41) LMNATP53HTTKCNH2CXCR3
SCHEMBL12735695 0.85 LMNA (0.41) LMNATP53HTTKCNH2CXCR3
SCHEMBL20365885 0.81 TP53 (0.55) LMNATP53HTTPSEN1PSEN2
SCHEMBL19098547 0.81 MC4R (0.39) SLC6A4PDE2A
SCHEMBL21725496 0.81 HTT (0.38) LMNATP53HTTPSEN1PSEN2
SCHEMBL19987472 0.81 KCNH2 (0.40) LMNATP53HTTKCNH2CXCR3
SCHEMBL23084281 0.80 LMNA (0.40) LMNATP53HTTKCNH2PSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230150998-A1 COMPOUNDS AS GLP-1R AGONISTS Terns, Inc. 2023-05-18 US disclosed
US-20210122757-A1 SPIROCYCLIC COMPOUNDS AS MODULATORS OF INDOLEAMINE 2,3-DIOXYGENASE Phenex Discovery Verwaltungs-GmbH (DE) 2021-04-29 US disclosed
US-10399932-B2 Inhibitors of indoleamine-2,3-dioxygenase for the treatment of cancer BRISTOL-MYERS SQUIBB COMPANY (US) 2019-09-03 US disclosed
US-20180079712-A1 INHIBITORS OF INDOLEAMINE-2,3-DIOXYGENASE FOR THE TREATMENT OF CANCER BRISTOL MYERS SQUIBB CO (US) 2018-03-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210122757-A1 SPIROCYCLIC COMPOUNDS AS MODULATORS OF INDOLEAMINE 2,3-DIOXYGENASE IDO1, IDO2, TPH1 LMNA 3679/4885TP53 4291/4885HTT 913/4885
US-10399932-B2 Inhibitors of indoleamine-2,3-dioxygenase for the treatment of cancer IDO1, IDO2, INMT LMNA 4373/4885TP53 352/4885HTT 3300/4885
US-20230150998-A1 COMPOUNDS AS GLP-1R AGONISTS GLP1R, GIPR, GCGR LMNA 2472/4885TP53 3988/4885HTT 780/4885
US-20180079712-A1 INHIBITORS OF INDOLEAMINE-2,3-DIOXYGENASE FOR THE TREATMENT OF CANCER IDO1, IDO2, INMT LMNA 4373/4885TP53 352/4885HTT 3300/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.