SCHEMBL19992736

SCHEMBL19992736

CCCCOC(=O)C1(c2cc(CN3CCN(C(=O)OC(C)(C)C)CC3)cc(C(F)(F)F)c2)CCCC1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 5/20 0.45
TSHR P16473 4/20 0.45
TACR1 P25103 1/20 0.43
ALDH1A1 P00352 2/20 0.42
USP2 O75604 7/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 2/20 0.41
MGLL Q99685 4/20 0.40
CYP3A4 P08684 6/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.38
CYP2C9 P11712 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19975519 0.89 CYP2D6 (0.51) CYP2D6TSHRTACR1ALDH1A1USP2
SCHEMBL19992929 0.81 CYP2D6 (0.45) CYP2D6TSHRTACR1ALDH1A1USP2
SCHEMBL28304786 0.77 CYP3A4 (0.47) CYP2D6TSHRTACR1ALDH1A1USP2
SCHEMBL20793838 0.77 MGLL (0.59) MGLL
SCHEMBL28304841 0.77 CYP2D6 (0.42) CYP2D6TSHRTACR1ALDH1A1USP2
SCHEMBL20151867 0.75 TSHR (0.58) CYP2D6TSHRTACR1ALDH1A1USP2
SCHEMBL20503443 0.75 CYP2D6 (0.50) CYP2D6TSHRTACR1ALDH1A1USP2
SCHEMBL20793596 0.75 ALDH1A1 (0.43) CYP2D6TSHRALDH1A1CYP1A2CYP3A4
SCHEMBL20137044 0.74 CYP2D6 (0.54) CYP2D6TSHRTACR1ALDH1A1USP2
SCHEMBL19974289 0.74 CYP2D6 (0.46) CYP2D6TSHRTACR1ALDH1A1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3515897-B1 PIPERAZINE CARBAMATES AS MODULATORS OF MAGL AND/OR ABHD6 AND THEIR USE H LUNDBECK AS (DK) 2021-08-18 EP disclosed
WO-2018053447-A1 PIPERAZINE CARBAMATES AND METHODS OF MAKING AND USING SAME ABIDE THERAPEUTICS, INC. (US) 2018-03-22 WO disclosed