SCHEMBL28304841

SCHEMBL28304841

CC(C)(C)OC(=O)C1(c2cc(CN3CCN(OC(=O)C(C)(C)C)CC3)cc(C(F)(F)F)c2)CCCC1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 6/20 0.42
TSHR P16473 5/20 0.42
USP2 O75604 8/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C19 P33261 2/20 0.42
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.39
CYP3A4 P08684 9/20 0.39
CYP2C9 P11712 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
GLA P06280 1/20 0.38
TACR1 P25103 1/20 0.37
HIF1A Q16665 1/20 0.37
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
MGLL Q99685 1/20 0.36
CASP1 P29466 1/20 0.36
CASP5 P51878 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19975519 0.87 CYP2D6 (0.51) CYP2D6TSHRUSP2CYP1A2CYP2C19
SCHEMBL28304786 0.85 CYP3A4 (0.47) CYP2D6TSHRUSP2CYP1A2CYP2C19
SCHEMBL28303890 0.78 TSHR (0.45) CYP2D6TSHRUSP2CYP1A2CYP2C19
SCHEMBL19992736 0.77 CYP2D6 (0.45) CYP2D6TSHRUSP2CYP1A2CYP2C19
SCHEMBL20769565 0.73 NOTUM (0.42) TACR1
SCHEMBL20769556 0.71 MGLL (0.61) MGLL
SCHEMBL29532670 0.71 MGLL (0.61) MGLL
SCHEMBL28303847 0.71 DDR1 (0.40) MEN1KMT2A
SCHEMBL19974449 0.71 MGLL (0.56) CYP2D6MGLL
SCHEMBL20769572 0.71 TACR1 (0.34) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109996790-A Piperazine carbamate and its preparation and application 阿比德治疗公司 2019-07-09 CN disclosed