Bromide

Bromide

SCHEMBL1999327

Br.CC(C)C(CN)C(C)C

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
TAAR1 Q96RJ0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1979 0.96
SCHEMBL4727402 0.92 ALDH1A1 (0.44) ALDH1A1TAAR1
Ammonia Solution, Strong SCHEMBL6136995 0.92 ALDH1A1 (0.44) ALDH1A1TAAR1
Fluoride SCHEMBL1025918 0.92 ALDH1A1 (0.44) ALDH1A1TAAR1
SCHEMBL3210302 0.92 ALDH1A1 (0.44) ALDH1A1TAAR1
Hydrochloric Acid SCHEMBL366444 0.92 ALDH1A1 (0.44) ALDH1A1TAAR1
Fluoride SCHEMBL73856 0.92 ALDH1A1 (0.44) ALDH1A1TAAR1
Trimethylammonium SCHEMBL4940105 0.86 ALDH1A1 (0.39) ALDH1A1
SCHEMBL4787789 0.86 ALDH1A1 (0.39) ALDH1A1
Dimethylamine SCHEMBL6889985 0.83 ALDH1A1 (0.37) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2920156-B9 PROCESS FOR THE PREPARATION OF MACROCYCLIC POLYAZACARBOXYLATE LIGANDS AND CHELATES GUERBET SA (FR) 2017-04-19 EP claimed
EP-2920156-B1 PROCESS FOR THE PREPARATION OF MACROCYCLIC POLYAZACARBOXYLATE LIGANDS AND CHELATES GUERBET SA (FR) 2016-12-07 EP claimed
US-11708345-B2 Continuous method for preparing carbonate esters UCHICAGO ARGONNE, LLC (US) 2023-07-25 US disclosed
CN-115335383-A Cyclic compound for organic electroluminescent device 默克专利有限公司 2022-11-11 CN disclosed
CN-110878057-B Method for preparing Raxinader 江苏宇田医药有限公司 2022-03-22 CN disclosed
US-20210276969-A1 CONTINUOUS METHOD FOR PREPARING CARBONATE ESTERS UCHICAGO ARGONNE, LLC (US) 2021-09-09 US disclosed
US-11028065-B1 Continuous method for preparing carbonate esters UCHICAGO ARGONNE, LLC (US) 2021-06-08 US disclosed
CN-110878057-A Method for preparing Raxinader 江苏宇田医药有限公司 2020-03-13 CN disclosed
EP-3037416-A1 PROCESS FOR SYNTHESIZING SUBSTITUTED ISOQUINOLINES Bristol-Myers Squibb Holdings Ireland (CH) 2016-06-29 EP disclosed
US-8877929-B2 Process for synthesizing substituted isoquinolines BRISTOL-MYERS SQUIBB COMPANY (US) 2014-11-04 US disclosed
US-20130123503-A1 Process for Synthesizing Substituted Isoquinolines BRISTOL-MYERS SQUIBB COMPANY (US) 2013-05-16 US disclosed
US-8207341-B2 Process or synthesizing substituted isoquinolines BRISTOL-MYERS SQUIBB COMPANY (US) 2012-06-26 US disclosed
EP-2326624-A2 PROCESS FOR SYNTHESIZING SUBSTITUTED ISOQUINOLINES Bristol-Myers Squibb Company (US) 2011-06-01 EP disclosed
WO-2010027889-A2 PROCESS FOR SYNTHESIZING SUBSTITUTED ISOQUINOLINES BRISTOL-MYERS SQUIBB COMPANY (US) 2010-03-11 WO disclosed
US-20100056792-A1 Process for Synthesizing Substituted Isoquinolines BRISTOL-MYERS SQUIBB COMPANY 2010-03-04 US disclosed
US-7417052-B2 Phenylene derivative having tetrazole ring or thiazolidinedione ring SANKYO COMPANY, LIMITED (JP) 2008-08-26 US disclosed
US-20070105846-A1 Phenylene derivative having tetrazole ring or thiazolidinedione ring RENASCIENCE CO., LTD (JP) 2007-05-10 US disclosed
EP-1679310-A1 PHENYLENE DERIVATIVE HAVING TETRAZOLE RING OR THIAZOLIDINEDIONE RING Sankyo Company, Limited (JP) 2006-07-12 EP disclosed
EP-0731797-A1 PARAMAGNETIC CHELATES FOR NUCLEAR MAGNETIC RESONANCE DIAGNOSIS BRACCO S.p.A. (IT) 1996-09-18 EP disclosed
WO-1995015319-A1 PARAMAGNETIC CHELATES FOR NUCLEAR MAGNETIC RESONANCE DIAGNOSIS BRACCO S.P.A. (IT) 1995-06-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100056792-A1 Process for Synthesizing Substituted Isoquinolines POLQ, SFPQ, SYNCRIP ALDH1A1 1643/4885TAAR1 3753/4885
US-11708345-B2 Continuous method for preparing carbonate esters CYP2E1, CYP2F1, CYP2C19 ALDH1A1 52/4885TAAR1 2080/4885
US-20130123503-A1 Process for Synthesizing Substituted Isoquinolines POLQ, SFPQ, SYNCRIP ALDH1A1 1643/4885TAAR1 3753/4885
US-11028065-B1 Continuous method for preparing carbonate esters CYP2E1, CYP2F1, CYP2C19 ALDH1A1 52/4885TAAR1 2080/4885
US-20210276969-A1 CONTINUOUS METHOD FOR PREPARING CARBONATE ESTERS CYP2E1, CYP2F1, CYP2C19 ALDH1A1 52/4885TAAR1 2080/4885
US-20070105846-A1 Phenylene derivative having tetrazole ring or thiazolidinedione ring JAK2, ABL1, CYP3A5 ALDH1A1 53/4885TAAR1 600/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.