SCHEMBL19993380

SCHEMBL19993380

N#Cc1ccc(-c2ccc(Cc3ccc(-c4ccc(C#N)c(I)c4)cc3)cc2)cc1I

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
RXRG P48443 1/20 0.40
AR P10275 3/20 0.37
PRKACA P17612 1/20 0.36
CDK8 P49336 1/20 0.36
CLK2 P49760 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
CDK9 P50750 1/20 0.36
CDK5 Q00535 1/20 0.36
PRKCQ Q04759 1/20 0.36
ROCK1 Q13464 1/20 0.36
DYRK1A Q13627 1/20 0.36
LRRK2 Q5S007 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
CYP11B1 P15538 10/20 0.35
CYP11B2 P19099 10/20 0.35
CYP17A1 P05093 6/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19993444 0.82 AR (0.33) RXRARXRBRXRGARCYP11B1
SCHEMBL21036112 0.81 MMP3 (0.47) ARCYP11B1CYP11B2PGRHRH3
SCHEMBL19993385 0.79 ESR1 (0.33) RXRARXRGCYP11B1CYP11B2CYP17A1
SCHEMBL19993333 0.75 S1PR1 (0.36) ARCYP11B1CYP11B2
SCHEMBL24108550 0.73 CYP11B1 (0.40) CYP11B1CYP11B2SNCA
SCHEMBL7143365 0.73 CYP11B1 (0.40) ARCYP11B1CYP11B2SNCA
SCHEMBL7135612 0.73 MAOB (0.38) SNCA
SCHEMBL19993384 0.73 CYP19A1 (0.33) RXRARXRBRXRGCYP11B1CYP11B2
SCHEMBL19993340 0.71 AR (0.32) ARPGR
SCHEMBL19993267 0.71 CYP17A1 (0.55) CYP11B1CYP11B2CYP17A1CYP19A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512920-B1 LIQUID CRYSTAL MEDIUM AND LIQUID CRYSTAL DEVICE MERCK PATENT GMBH (DE) 2020-11-04 EP disclosed
WO-2018050573-A1 LIQUID CRYSTAL MEDIUM AND LIQUID CRYSTAL DEVICE MERCK PATENT GMBH (DE) 2018-03-22 WO disclosed