SCHEMBL19994153

SCHEMBL19994153

O=c1[nH]c(=O)n(CC(F)(F)F)c2sccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 2/20 0.36
ERCC5 P28715 2/20 0.36
FEN1 P39748 2/20 0.36
ERCC4 Q92889 2/20 0.36
PARP1 P09874 3/20 0.35
PARP15 Q460N3 2/20 0.35
TNKS2 Q9H2K2 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 2/20 0.35
TNKS O95271 1/20 0.35
MEN1 O00255 1/20 0.35
MAPK1 P28482 1/20 0.35
GRIK1 P39086 1/20 0.34
GRIA1 P42261 1/20 0.34
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
HTR2A P28223 1/20 0.33
PDE1B Q01064 1/20 0.33
DAO P14920 1/20 0.33
BRD4 O60885 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31751098 0.79 GRIK1 (0.38) ERCC1ERCC5FEN1ERCC4PARP1
SCHEMBL6670689 0.76 ALDH1A1 (0.40) ERCC1ERCC5FEN1ERCC4PARP15
SCHEMBL2980047 0.71 ALDH1A1 (0.54) ERCC1ERCC5FEN1ERCC4PARP1
SCHEMBL2987031 0.70 PARP15 (0.41) ERCC1ERCC5FEN1ERCC4PARP1
SCHEMBL7507593 0.70 DAO (0.53) ERCC1ERCC5FEN1ERCC4PARP1
SCHEMBL31257840 0.66 TNKS2 (0.45) ERCC1ERCC5FEN1ERCC4PARP1
SCHEMBL8141804 0.66 PARP1 (0.40) ERCC1ERCC5FEN1ERCC4PARP1
SCHEMBL116024 0.64 METAP2 (0.39) ERCC1ERCC5FEN1ERCC4ALDH1A1
SCHEMBL6242682 0.62 CYP1A2 (0.64) ERCC1ERCC5FEN1ERCC4KMT2A
SCHEMBL4175626 0.61 MEN1 (0.62) KMT2AALDH1A1MEN1MAPK1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3515919-A1 N3-CYCLICALLY SUBSTITUTED THIENOURACILES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2019-07-31 EP disclosed
WO-2018054846-A1 N3-CYCLICALLY SUBSTITUTED THIENOURACILES AND USE THEREOF BAYER AKTIENGESELLSCHAFT (DE) 2018-03-29 WO disclosed