SCHEMBL19997239

SCHEMBL19997239

CC(C)S(=O)(=O)Nc1ccccc1C(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.54
MEN1 O00255 2/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
TSHR P16473 1/20 0.54
CYP2C19 P33261 1/20 0.54
GAA P10253 1/20 0.52
POLB P06746 4/20 0.47
MAPK1 P28482 1/20 0.47
SLC22A12 Q96S37 5/20 0.46
ALDH1A1 P00352 4/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
BCL2L1 Q07817 1/20 0.45
MCL1 Q07820 1/20 0.45
LMNA P02545 1/20 0.44
RXFP1 Q9HBX9 1/20 0.43
HPGD P15428 1/20 0.43
NR3C1 P04150 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16492688 0.80 KMT2A (0.58) KMT2AMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL13565375 0.79 SCD (0.43) KMT2AMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL21104478 0.79 MCL1 (0.40) KMT2AMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL10116480 0.78 SMN1; SMN2 (0.59) GAAPOLBMAPK1ALDH1A1LMNA
SCHEMBL22455897 0.78 SLC22A12 (0.49) SLC22A12NR3C1
SCHEMBL19303635 0.77 PSIP1 (0.61) KMT2AMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL20290538 0.77 KMT2A (0.55) KMT2AMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL14830619 0.77 PSIP1 (0.59) KMT2AMEN1TSHRGAAPOLB
SCHEMBL13564954 0.75 GRIA1 (0.50) KMT2AMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL13469116 0.75 ALDH1A1 (0.50) KMT2AMEN1TSHRGAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9926309-B2 Pi-kinase inhibitors with anti-infective activity THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2018-03-27 US disclosed