SCHEMBL19997252

SCHEMBL19997252

CCCC(CC)C(=O)c1nn(C)c2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.52
TSHR P16473 2/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.44
HTR3E A5X5Y0 2/20 0.43
HTR3B O95264 2/20 0.43
HTR3A P46098 2/20 0.43
HTR3D Q70Z44 2/20 0.43
HTR3C Q8WXA8 2/20 0.43
SLC22A2 O15244 1/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA4 P43681 1/20 0.43
KCNH2 Q12809 1/20 0.43
SLC47A1 Q96FL8 1/20 0.43
RBP4 P02753 1/20 0.40
ELANE P08246 3/20 0.40
F2 P00734 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19997287 0.84 HTR4 (0.48) CYP3A4KCNH2HTR2A
SCHEMBL25139488 0.82 KDM4E (0.59) KDM4ETSHRALDH1A1CYP3A4MAPK1
SCHEMBL20250836 0.78 CNR1 (0.47) KDM4ETSHRHSD17B10HTR3AELANE
SCHEMBL17321382 0.78 KDM4E (0.66) KDM4ETSHRALDH1A1CYP3A4MAPK1
SCHEMBL19902669 0.77 KDM4E (0.56) KDM4ETSHRALDH1A1CYP3A4MAPK1
SCHEMBL19902668 0.75 KDM4E (0.57) KDM4ETSHRALDH1A1CYP3A4MAPK1
SCHEMBL496589 0.73 KDM4E (0.62) KDM4ETSHRALDH1A1CYP3A4MAPK1
SCHEMBL30251861 0.73 KDM4E (0.62) KDM4ETSHRALDH1A1CYP3A4MAPK1
SCHEMBL30467838 0.73 KDM4E (0.62) KDM4ETSHRALDH1A1CYP3A4MAPK1
SCHEMBL7297926 0.73 KDM4E (0.62) KDM4ETSHRALDH1A1CYP3A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9926282-B2 Phthalazinones and isoquinolinones as rock inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2018-03-27 US disclosed