SCHEMBL20000896

SCHEMBL20000896

COc1ccc2cc(-c3n[nH]cc3OC)ccc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 2/20 0.50
HSD17B2 P37059 2/20 0.50
NPC1 O15118 4/20 0.49
RAB9A P51151 4/20 0.49
CYP11B2 P19099 9/20 0.47
CYP11B1 P15538 8/20 0.47
CYP1A2 P05177 4/20 0.47
CYP3A4 P08684 3/20 0.47
CYP2C9 P11712 3/20 0.47
GSTP1 P09211 1/20 0.47
NISCH Q9Y2I1 1/20 0.47
CYP17A1 P05093 3/20 0.45
CYP19A1 P11511 1/20 0.45
CASP3 P42574 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
CYP2A6 P11509 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CYP2D6 P10635 2/20 0.42
CYP2C19 P33261 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12788907 0.86 HSD17B1 (0.43) HSD17B1HSD17B2NPC1RAB9ACYP11B2
SCHEMBL12846896 0.79 CYP11B1 (0.52) HSD17B1HSD17B2NPC1RAB9ACYP11B2
SCHEMBL11723032 0.74 HSD17B1 (0.83) HSD17B1HSD17B2NPC1RAB9ACYP11B2
SCHEMBL12051687 0.74 HSD17B1 (0.83) HSD17B1HSD17B2NPC1RAB9ACYP11B2
SCHEMBL27912509 0.72 HSD17B1 (0.66) HSD17B1HSD17B2CYP11B2CYP11B1CYP1A2
SCHEMBL11620293 0.72 ALDH1A1 (0.46) NPC1RAB9A
SCHEMBL12318102 0.71 ITK (0.67) NPC1RAB9ACYP11B2CYP11B1CYP1A2
SCHEMBL14041533 0.70 HSD17B1 (0.76) HSD17B1HSD17B2NPC1RAB9ACYP11B2
SCHEMBL22106285 0.70 HSD17B1 (0.76) HSD17B1HSD17B2NPC1RAB9ACYP11B2
SCHEMBL3020390 0.70 HSD17B1 (0.76) HSD17B1HSD17B2NPC1RAB9ACYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2291358-B1 GLUCAGON RECEPTOR ANTAGONISTS, COMPOSITIONS, AND METHODS FOR THEIR USE MERCK SHARP & DOHME (US) 2018-03-28 EP disclosed