SCHEMBL20001577

SCHEMBL20001577

CCc1ccnc(N)c1C

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 8/20 0.56
NOS3 P29474 7/20 0.56
NOS1 P29475 4/20 0.41
PRKCI P41743 1/20 0.36
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ROCK1 Q13464 1/20 0.35
TLR8 Q9NR97 1/20 0.35
DHFR P00374 1/20 0.34
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14035774 0.83 NOS2 (0.46) NOS2NOS3NOS1PRKCIROCK1
SCHEMBL31032970 0.81 NOS2 (0.54) NOS2NOS3NOS1KDM4EMEN1
SCHEMBL23012667 0.81 NOS2 (0.54) NOS2NOS3NOS1KDM4EMEN1
SCHEMBL15528179 0.80 NOS2 (0.49) NOS2NOS3NOS1TLR8
SCHEMBL3264472 0.80 NOS2 (0.52) NOS2NOS3NOS1PRKCITLR8
SCHEMBL357771 0.78 NOS2 (0.64) NOS2NOS3NOS1PRKCITLR8
SCHEMBL26105660 0.78 NOS2 (0.50) NOS2NOS3NOS1KDM4EMEN1
SCHEMBL27804907 0.78 NOS2 (0.50) NOS2NOS3NOS1PRKCIKDM4E
SCHEMBL21806239 0.77 NOS2 (0.46) NOS2NOS3KDM4EMEN1KMT2A
SCHEMBL3801869 0.77 NOS2 (0.38) NOS2NOS3NOS1PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563043-A SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 葛兰素史密斯克莱知识产权发展有限公司 2019-04-02 CN disclosed
WO-2018057810-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS GILEAD SCIENCES, INC. (US) 2018-03-29 WO disclosed