SCHEMBL20001657

SCHEMBL20001657

N#Cc1ccc2[nH]c(-c3ccc(N4CCOCC4)cc3)nc2c1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RHEB Q15382 1/20 0.50
SIRT2 Q8IXJ6 1/20 0.48
SIRT1 Q96EB6 1/20 0.48
PKN1 Q16512 1/20 0.47
PKN2 Q16513 1/20 0.47
PARP1 P09874 1/20 0.47
CBFB Q13951 1/20 0.46
TBK1 Q9UHD2 6/20 0.45
LRRK2 Q5S007 1/20 0.45
JAK2 O60674 1/20 0.45
CHEK2 O96017 2/20 0.45
ACHE P22303 1/20 0.45
CHEK1 O14757 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30343715 1.00 RHEB (0.50) RHEBSIRT2SIRT1PKN1PKN2
SCHEMBL30343735 0.89 RHEB (0.51) RHEBSIRT2SIRT1PKN1PKN2
SCHEMBL19994743 0.89 RHEB (0.51) RHEBSIRT2SIRT1PKN1PKN2
SCHEMBL1664192 0.87 ALDH1A1 (0.53) SIRT2SIRT1LRRK2CHEK2
SCHEMBL1663221 0.81 PARP1 (0.52) SIRT2SIRT1PARP1CBFBCHEK2
SCHEMBL8772505 0.81 SIRT2 (0.59) SIRT2SIRT1CBFBCHEK2ACHE
SCHEMBL1666722 0.81 KDM4E (0.50) SIRT2SIRT1PARP1CBFBCHEK2
SCHEMBL8768585 0.80 CHEK2 (0.56) SIRT2SIRT1LRRK2CHEK2
SCHEMBL8769224 0.80 CHEK2 (0.56) SIRT2SIRT1LRRK2CHEK2
SCHEMBL19994744 0.80 PKN1 (0.61) RHEBSIRT2SIRT1PKN1PKN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12509465-B2 Benzoimidazole derivatives as anticancer agents CENTRE LEON BERARD (FR) 2025-12-30 US disclosed
EP-3515904-B1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2024-01-17 EP disclosed
EP-3515904-B1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2024-01-17 EP disclosed
CN-110234640-B Benzimidazole derivatives as anticancer agents 利昂贝拉尔中心 2023-04-07 CN disclosed
US-20220348587-A1 Benzoimidazole Derivatives As Anticancer Agents CENTRE LEON BERARD (FR) 2022-11-03 US disclosed
US-20220348587-A1 Benzoimidazole Derivatives As Anticancer Agents CENTRE LEON BERARD (FR) 2022-11-03 US disclosed
US-11384081-B2 Benzoimidazole derivatives as anticancer agents CENTRE LEON BERARD (FR) 2022-07-12 US disclosed
US-11384081-B2 Benzoimidazole derivatives as anticancer agents CENTRE LEON BERARD (FR) 2022-07-12 US disclosed
US-20210292328-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2021-09-23 US disclosed
US-20210292328-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2021-09-23 US disclosed
WO-2018054989-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2018-03-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12509465-B2 Benzoimidazole derivatives as anticancer agents CCAR2, MAPKAP1, BCOR RHEB 500/4885SIRT2 1935/4885SIRT1 2148/4885
US-20210292328-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS TMBIM6, BAX, MAPK14 RHEB 798/4885SIRT2 1954/4885SIRT1 2241/4885
US-11384081-B2 Benzoimidazole derivatives as anticancer agents TMBIM6, BAX, MAPK14 RHEB 798/4885SIRT2 1954/4885SIRT1 2241/4885
US-20220348587-A1 Benzoimidazole Derivatives As Anticancer Agents TMBIM6, BAX, BCL2 RHEB 839/4885SIRT2 1990/4885SIRT1 2253/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.