SCHEMBL19994744

SCHEMBL19994744

N#Cc1ccc2nc(-c3ccc(N4CCCCC4)cc3)[nH]c2c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKN1 Q16512 1/20 0.61
PKN2 Q16513 1/20 0.61
NPBWR1 P48145 1/20 0.60
CHEK2 O96017 3/20 0.57
SIRT2 Q8IXJ6 1/20 0.55
SIRT1 Q96EB6 1/20 0.55
DGAT1 O75907 2/20 0.52
SOAT1 P35610 2/20 0.52
KCNH2 Q12809 2/20 0.52
RHEB Q15382 1/20 0.51
TOP1 P11387 2/20 0.48
TOP2A P11388 2/20 0.48
ALDH1A1 P00352 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
HPGD P15428 1/20 0.48
HSD17B10 Q99714 1/20 0.48
METAP2 P50579 1/20 0.48
METAP1 P53582 1/20 0.48
AURKA O14965 1/20 0.48
ACHE P22303 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30343735 0.90 RHEB (0.51) PKN1PKN2NPBWR1CHEK2SIRT2
SCHEMBL19994743 0.90 RHEB (0.51) PKN1PKN2NPBWR1CHEK2SIRT2
SCHEMBL20982510 0.84 PKN1 (0.82) PKN1PKN2CHEK2DGAT1SOAT1
SCHEMBL20001657 0.80 RHEB (0.50) PKN1PKN2CHEK2SIRT2SIRT1
SCHEMBL30343715 0.80 RHEB (0.50) PKN1PKN2CHEK2SIRT2SIRT1
SCHEMBL19175759 0.78 DGAT1 (0.77) NPBWR1SIRT2SIRT1DGAT1SOAT1
SCHEMBL3341423 0.78 PKN1 (0.72) PKN1PKN2NPBWR1CHEK2DGAT1
SCHEMBL14816640 0.78 PKN1 (0.72) PKN1PKN2CHEK2SIRT2DGAT1
SCHEMBL18764054 0.77 CHEK2 (0.78) PKN1PKN2NPBWR1CHEK2DGAT1
SCHEMBL902210 0.77 PKN1 (0.60) PKN1PKN2CHEK2DGAT1SOAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3515904-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS Centre Leon Berard (FR) 2019-07-31 EP disclosed
WO-2018054989-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2018-03-29 WO disclosed