SCHEMBL20002025

SCHEMBL20002025

COc1ccc(OC(C)(C(F)(F)F)C(F)(F)F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA7 P43166 2/20 0.50
CA9 Q16790 2/20 0.50
CA12 O43570 1/20 0.50
CA14 Q9ULX7 1/20 0.50
PDK1 Q15118 1/20 0.43
PDK2 Q15119 1/20 0.43
PDK3 Q15120 1/20 0.43
PDK4 Q16654 1/20 0.43
ACHE P22303 1/20 0.42
HSD11B1 P28845 1/20 0.42
TDP1 Q9NUW8 4/20 0.41
MAPK1 P28482 3/20 0.41
GAA P10253 2/20 0.40
MAPT P10636 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002023 0.82 GAA (0.40) ACHEHSD11B1TDP1GAAMAPT
SCHEMBL19477798 0.81 CA1 (0.55) CA1CA2CA7CA9CA12
SCHEMBL20003172 0.79 CA4 (0.40) PDK1PDK2PDK3PDK4MAPK1
SCHEMBL514500 0.78 CA1 (0.58) CA1CA2CA7CA9CA12
SCHEMBL20714605 0.77 CA1 (0.50) CA1CA2CA7CA9CA12
SCHEMBL9324454 0.76 CA1 (0.55) CA1CA2CA7CA9CA12
SCHEMBL5285766 0.75 CA1 (0.61) CA1CA2CA7CA9CA12
SCHEMBL1246270 0.73 CA1 (0.50) CA1CA2CA7CA9CA12
SCHEMBL9171548 0.73 CA1 (0.50) CA1CA2CA7CA9CA12
SCHEMBL2084265 0.73 KIF11 (0.53) CA1CA2CA7CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed